Glycoside

GD002534
Name:
CALICHEAMICIN BETA1 BRFormula:
C56H76O21N3S4BrSmiles:
COC(=O)NC1=C2C(=CCSSSC)[C@](O)(C#CC=CC#CC2OC2OC(C)C(NOC3CC(O)C(SC(=O)c4c(C)c(Br)c(OC5OC(C)C(O)C(OC)C5O)c(OC)c4OC)C(C)O3)C(O)C2OC2CC(OC)C(NC(C)C)CO2)CC1=OAglycone:
COC(=O)NC1=C2C(=CCSSSC)C(O)(C#CC=CC#CC2O)CC1=O.COC1CC(O)OCC1NC(C)C.COc1c(O)c(Br)c(C)c(C(=O)SC2C(O)CC(ON)OC2C)c1OCSugarmoiety:
CC1OC(O)C(O)C(O)C1O.COC1C(O)C(C)OC(O)C1OOther Identifiers
Properties
HBA: | 24 | RingCount: | 7 |
HBD: | 8 | FractionCSP3: | 0.66 |
AlogP: | 3.74 | Num_rotatable_bonds: | 22 |
MolWt: | 1335.4 | Num_heavy_atoms: | 85 |
TPSA: | 308.44 | NumAromaticRings: | 1 |
Unique Aglycone
AD01088
Formula: C18H17O5NS3
Smiles:
COC(=O)NC1=C2C(=CCSSSC)C(O)(C#CC=CC#CC2O)CC1=OHBA: | 6 | RingCount: | 2 |
HBD: | 3 | FractionCSP3: | 0.33 |
AlogP: | 1.82 | Num_rotatable_bonds: | 5 |
MolWt: | 423.54 | Num_heavy_atoms: | 27 |
TPSA: | 95.86 | NumAromaticRings: | 0 |
AD02411
Formula: C9H19O3N
Smiles:
COC1CC(O)OCC1NC(C)CHBA: | 4 | RingCount: | 1 |
HBD: | 2 | FractionCSP3: | 1.0 |
AlogP: | 0.11 | Num_rotatable_bonds: | 3 |
MolWt: | 189.26 | Num_heavy_atoms: | 13 |
TPSA: | 50.72 | NumAromaticRings: | 0 |
AD02412
Formula: C16H22O7NSBr
Smiles:
COc1c(O)c(Br)c(C)c(C(=O)SC2C(O)CC(ON)OC2C)c1OCHBA: | 8 | RingCount: | 2 |
HBD: | 4 | FractionCSP3: | 0.56 |
AlogP: | 2.11 | Num_rotatable_bonds: | 5 |
MolWt: | 452.32 | Num_heavy_atoms: | 26 |
TPSA: | 120.47 | NumAromaticRings: | 1 |